Bioactivity:

Olcegepant is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP).

CAS nr:

204697-65-4

Purity:

98%

Molecular Weight:

869,65

SMILES:

NCCCC[C@@H](C(N(CC1)CCN1c1ccncc1)=O)NC([C@@H](Cc(cc1Br)cc(Br)c1O)NC(N(CC1)CCC1N(Cc(cccc1)c1N1)C1=O)=O)=O

Formula:

C38H47Br2N9O5

Pathway:

Membrane transporter/Ion channel

Target:

CGRP Receptor