Bioactivity:

BRD7389 is an inducer of insulin expression in pancreatic _-cells and a specific inhibitor of RSK family kinase (IC50s: 1.5 _M, 2.4 _M, and 1.2 _M for RSK1, RSK2, and RSK3).

CAS nr:

376382-11-5

Purity:

98%

Molecular Weight:

366,41

SMILES:

O=C(C(C=CC=C1)=C1C2=C(NCCC3=CC=CC=C3)C(N4)=O)C5=C2C4=CC=C5

Formula:

C24H18N2O2

Pathway:

PI3K/Akt/mTOR signaling,MAPK,Cell Cycle/Checkpoint

Target:

S6 Kinase,S6 Kinase,CDK