CK2/ERK8-IN-1 T10827
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
CK2/ERK8-IN-1 is a dual inhibitor of casein kinase 2 (CK2) (Ki: 0.25 ᄉM) and ERK8 (IC50s: 0.50 _M) with pro-apoptotic efficacy. CK2/ERK8-IN-1 also binds to PIM1, DYRK1A, and HIPK2 (Kis: 8.65 ᄉM, 11.9 ᄉM, and 15.25 ᄉM).
CAS nr:
1085822-09-8
Purity:
98%
Molecular Weight:
534,82
SMILES:
O=C(O)CN1C2=C(Br)C(Br)=C(Br)C(Br)=C2N=C1N(C)C
Formula:
C11H9Br4N3O2
Pathway:
Metabolism,Stem Cells
Target:
Casein Kinase,Casein Kinase
