JAK1-IN-4 T15606
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
JAK1-IN-4 is a selective JAK1 inhibitor (IC50s: 85 nM, 12.8 _M and >30 _M for JAK1, JAK2, and JAK3, respectively). JAK1-IN-4 inhibits STAT3 phosphorylation in NCI-H 1975 cells (IC50, 227 nM).
CAS nr:
2091134-35-7
Purity:
98%
Molecular Weight:
521,59
SMILES:
O=C(NC1=CC=CC2=C1NC=C2C3=C(C=NC(NC4=CN(N=C4OC)C)=N3)F)[C@H](N5CCN([C@@H](C5)C)C)C
Formula:
C26H32FN9O2
Pathway:
JAK/STAT signaling,Chromatin/Epigenetic,Stem Cells,Angiogenesis
Target:
JAK,JAK,JAK,JAK
