Bioactivity:

CB1 inverse agonist 1 is an orally active, and specific inverse agonist of the CB1 receptor (IC50s: 7.5 nM and 4100 nM for CB1 and CB2 receptors) with anorexigenic effects.

CAS nr:

852315-00-5

Purity:

98%

Molecular Weight:

514,79

SMILES:

CC(NC1=C(C(C)=O)C(N(C)C2=NC(C3=CC=C(Cl)C=C3Cl)=C(C4=CC=C(Cl)C=C4)C=C12)=O)=O

Formula:

C25H18Cl3N3O3

Pathway:

GPCR/G Protein

Target:

Cannabinoid Receptor