Bioactivity:

UNC 0646 is a potent and selective inhibitor of the homologous protein lysine methyltransferases, G9a and GLP (IC50s: 6 nM/15 nM for G9a/GLP). UNC0646 potently blocks G9a/GLP methyltransferase activity in cells (IC50: 10 nM in MCF7 cells); exhibits low ce

CAS nr:

1320288-17-2

Purity:

98%

Molecular Weight:

621,9

SMILES:

COC1=C(OCCCN2CCCCC2)C=C2N=C(N=C(NC3CCN(CC3)C3CCCCC3)C2=C1)N1CCCN(CC1)C(C)C

Formula:

C36H59N7O2

Pathway:

Chromatin/Epigenetic

Target:

Histone Methyltransferase