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GSK180736A T3513

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Specifications

size	1mg/5mg/10mg/25mg/50mg/100mg

Bioactivity:

GSK180736A is an effective and selective GRK2 inhibitor (IC50: 0.77 _M) and >100-fold selectivity over other GRKs. It is a weak inhibitor of PKA (IC50: 30 _M), but highly effective against ROCK1 (IC50: 100 nM).

CAS nr:

817194-38-0

Purity:

98%

Molecular Weight:

365,13

SMILES:

CC1=C(C(NC(=O)N1)c1ccc(cc1)F)C(=O)Nc1cc2c(cc1)[nH]nc2

Formula:

C19H16FN5O2

Pathway:

Tyrosine Kinase/Adaptors,Cell Cycle/Checkpoint,Stem Cells,Cytoskeletal Signaling,GPCR/G Protein

Target:

PKA,ROCK,ROCK,ROCK,GRK