Bioactivity:

GS-6201 is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors (Ki: 22 nM). GS-62013 attenuates the airway reactivity induced by NECA, AMP, or allergen in sensitized mice.

CAS nr:

752222-83-6

Purity:

98%

Molecular Weight:

446,43

SMILES:

O=C(N(CCC)C1=O)N(CC)C(C1=N2)=NC2C3=CN(N=C3)CC4=CC=CC(C(F)(F)F)=C4

Formula:

C21H21F3N6O2

Pathway:

Neuroscience,GPCR/G Protein

Target:

Adenosine Receptor,Adenosine Receptor