Bioactivity:

NNC052090 is a GABA uptake inhibitor that displays moderate selectivity for BGT-1 transporters with Ki values are 1.4, 15, 19 and 41 _M for hBGT-1, hGAT-3, hGAT-1 and hGAT-2 respectively. NNC052090 also displays affinity at _1- and D2-receptors with IC50

CAS nr:

184845-43-0

Purity:

98%

Molecular Weight:

414,55

SMILES:

OC1(C2=CC=CC=C2OC)CCN(CCCN3C4=C(C5=C3C=CC=C5)C=CC=C4)CC1

Formula:

C27H30N2O2

Pathway:

Target: