Bioactivity:

4SC-202 is a selective class I HDAC inhibitor with IC50 of 1.20 _M, 1.12 _M, and 0.57 _M for HDAC1, HDAC2, and HDAC3, respectively. Also displays inhibitory activity against Lysine specific demethylase 1 (LSD1). Phase 1.

CAS nr:

910462-43-0

Purity:

98%

Molecular Weight:

447,51

SMILES:

Cn1cc(cn1)-c1ccc(cc1)S(=O)(=O)n1ccc(\C=C\C(=O)Nc2ccccc2N)c1

Formula:

C23H21N5O3S

Pathway:

DNA Damage/DNA Repair,Chromatin/Epigenetic,Apoptosis

Target:

HDAC,HDAC,Apoptosis