(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin TP2136
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
Selective vasopressin V1A receptor antagonist. Inhibits vasopressin and oxytocin-induced increases in intracellular calcium concentrations in vitro (IC50 values are 5 and 30 nM respectively). Exhibits potent and prolonged antivasopressor activity and indu
CAS nr:
73168-24-8
Purity:
98%
Molecular Weight:
1151,38
SMILES:
Formula:
C52H74N14O12S2
Pathway:
Target:
