Bioactivity:

GSK2807 Trifluoroacetate is a selective and SAM-competitive inhibitor of SMYD3 (Ki: 14 nM; IC50: 130 nM).

CAS nr:

2245255-66-5

Purity:

98%

Molecular Weight:

566,53

SMILES:

NC1=C2C(N([C@H]3[C@H](O)[C@H](O)[C@@H](CN(CC[C@H](N)C(O)=O)CCCN(C)C)O3)C=N2)=NC=N1.OC(C(F)(F)F)=O

Formula:

C21H33F3N8O7

Pathway:

Chromatin/Epigenetic

Target:

Histone Methyltransferase