Bioactivity:

PKC-IN-1 is a ATP-competitive and reversible conventional PKC enzymes inhibitor (PKC_, PKC_I, PKC_II, PKC_, PKC_, PKC mu and PKC_ with IC50s of 2.3, 8.1, 7.6, 25.6, 57.5, 314, 808 nM , respectively).

CAS nr:

1046787-18-1

Purity:

98%

Molecular Weight:

500,61

SMILES:

O=C(N1[C@@H](C)CN(CC2CCOCC2)[C@H](C)C1)N(C3)C(C)(C)C4=C3C(NC5=NC(C)=NC=C5F)=NN4

Formula:

C25H37FN8O2

Pathway:

Cytoskeletal Signaling,Chromatin/Epigenetic

Target:

PKC,PKC