Bioactivity:

CF53 is a highly potent, selective, and orally active inhibitor of BET protein (Ki: <1 nM, Kd: 2.2 nM, IC50: 2 nM for BRD4 BD1).

CAS nr:

1808160-52-2

Purity:

98%

Molecular Weight:

443,5

SMILES:

COC1=C(C2=C(C)ON=C2C)C=C(NC3=C4C(NC5=CC(C6CC6)=NN5C)=NC(C)=N3)C4=C1

Formula:

C24H25N7O2

Pathway:

Chromatin/Epigenetic

Target:

Epigenetic Reader Domain