Bioactivity:

(R)-Elagolix is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively.�administered orally, that unlike injectable depot GnRH agonists and antagonists, produces a dose-dependent suppression of ovarian estrogen pr

CAS nr:

834153-87-6

Purity:

98%

Molecular Weight:

631,59

SMILES:

CC1=C(C(=O)N(C(=O)N1CC2=C(C=CC=C2F)C(F)(F)F)C[C@@H](C3=CC=CC=C3)NCCCC(=O)O)C4=C(C(=CC=C4)OC)F

Formula:

C32H30F5N3O5

Pathway:

GPCR/G Protein

Target:

GNRH Receptor