Bioactivity:

MS023 is a potent, selective, and cell-active Type I PRMT inhibitor with IC50 of 30 nM, 119 nM, 83 nM, 4 nM, and 5 nM for PRMT1, PRMT3, PRMT4, PRMT6 and PRMT8, respectively.

CAS nr:

1831110-54-3

Purity:

98%

Molecular Weight:

287,4

SMILES:

C(CN)N(C)Cc1c[nH]cc1c1ccc(cc1)OC(C)C

Formula:

C17H25N3O

Pathway:

Chromatin/Epigenetic

Target:

Histone Methyltransferase