Bioactivity:

VU6005806 is a potent positive allosteric modulator (PAM) of muscarinic acetylcholine receptor subtype 4 (M4) (EC50s: 94 nM, 28 nM, 87 nM, and 68 nM for human, rat, dog, and cyno M4, respectively), and used in the study of neuropsychiatric disorders.

CAS nr:

2180914-37-6

Purity:

98%

Molecular Weight:

439,41

SMILES:

NC1=C(C(NC2CN(C3=NC=C(C(F)(F)F)C=N3)C2)=O)SC4=NN=C(OC)C(C)=C41

Formula:

C17H16F3N7O2S

Pathway:

Others

Target:

Others