Bioactivity:

ARP-100 is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM). ARP-100 shows the less inhibitory activity towards MMP-1 (>50 _M), MMP-3 (4.5 _M), MMP-7 (>50 _M), and MMP-9 (0.2 _M)[1][2]. ARP-100 interacts with S1_ pocket of MMP-

CAS nr:

704888-90-4

Purity:

98%

Molecular Weight:

364,42

SMILES:

CC(C)ON(CC(NO)=O)S(c(cc1)ccc1-c1ccccc1)(=O)=O

Formula:

C17H20N2O5S

Pathway:

Proteases/Proteasome

Target:

MMP