Bioactivity:

Ogerin is a selective GPR68 positive allosteric modulator (pEC50: 6.83). Ogerin blocks recall in fear conditioning in mice. Ogerin displays inverse agonist and antagonist activity (Ki, 220 nM) at A2A receptor and weak antagonist activity (Ki, 736 nM) at 5

CAS nr:

1309198-71-7

Purity:

98%

Molecular Weight:

307,35

SMILES:

OCC1=C(C2=NC(N)=NC(NCC3=CC=CC=C3)=N2)C=CC=C1

Formula:

C17H17N5O

Pathway:

GPCR/G Protein,Neuroscience,Neuroscience,GPCR/G Protein,Others

Target:

5-HT Receptor,5-HT Receptor,Adenosine Receptor,Adenosine Receptor,Others