Bioactivity:

Brilaroxazine (RP5603) is a partial agonist of dopamine (DA) D2, D3, and D4 receptors, 5-HT1A (Ki: 1.5 nM) and 5-HT2A (Ki: 2.5 nM), and has antagonist activity at 5-HT2B (Ki: 0.19 nM), and 5-HT7 (Ki: 2.7 nM) receptors.

CAS nr:

1239729-06-6

Purity:

98%

Molecular Weight:

450,36

SMILES:

O=C1NC2=CC(OCCCCN3CCN(C(C=CC=C4Cl)=C4Cl)CC3)=CC=C2OC1

Formula:

C22H25Cl2N3O3

Pathway:

GPCR/G Protein,Neuroscience,GPCR/G Protein,Neuroscience

Target:

5-HT Receptor,5-HT Receptor,Dopamine Receptor,Dopamine Receptor