Bioactivity:

DG-041 is an antagonist of high-affinity EP3 receptor (IC50s: 4.6 nM and 8.1 nM in the binding and FLIPR assay, respectively). DG-041 inhibits PGE2 facilitation of platelet aggregation and has the blood-brain barrier permeability.

CAS nr:

861238-35-9

Purity:

98%

Molecular Weight:

592,32

SMILES:

O=C(NS(=O)(C1=CC(Cl)=C(Cl)S1)=O)/C=C/C2=CC(F)=CC3=C2N(CC4=CC=C(Cl)C=C4Cl)C=C3C

Formula:

C23H15Cl4FN2O3S2

Pathway:

Others

Target:

Others