Bioactivity:

AC-178335 is a pure somatostatin (SRIF) antagonist with an affinity constant (Ki) of 172 +/- 12 nM. AC-178335 blocks SRIF inhibition of adenylate cyclase in vitro (IC50 = 5.1 +/- 1.4 microM). It induces GH release when given alone (50 micrograms intraveno

CAS nr:

212966-15-9

Purity:

98%

Molecular Weight:

946,13

SMILES:

CC[C@@H](C)[C@@H](NC([C@H](NC([C@H](NC(C)=O)CC1=CNC=N1)=O)CC2=CC=CC=C2)=O)C(N[C@H](CCCNC(N)=N)C(N[C@H](CC3=CNC4=C3C=CC=C4)C(N[C@H](CC5=CC=CC=C5)C(N)=O)=O)=O)=O

Formula:

C49H63N13O7

Pathway:

Target: