Bioactivity:

GSK3368715�is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50s: 3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8)).�It has strong

CAS nr:

1629013-22-4

Purity:

98%

Molecular Weight:

366,54

SMILES:

CNCCN(CC1=CNN=C1C2CCC(COCC)(COCC)CC2)C

Formula:

C20H38N4O2

Pathway:

Chromatin/Epigenetic

Target:

Histone Methyltransferase