Bioactivity:

PDK1-IN-RS2 inhibits the activation of the downstream kinases S6K1 by PDK1. PDK1-IN-RS2 is a mimic of the peptide docking motif (PIFtide) and is a substrate-selective PDK1 inhibitor (Kd: 9 _M).

CAS nr:

1643958-89-7

Purity:

98%

Molecular Weight:

380,89

SMILES:

O=S(C1=CC2=CC=CC=C2S1)(NC3=NC4=CC=C(C=C4S3)Cl)=O

Formula:

C15H9ClN2O2S3

Pathway:

PI3K/Akt/mTOR signaling

Target:

PDK