Bioactivity:

PROTAC BRD4 Degrader-1 is an efficacious degrader of BRD4(BRD4 BD1,IC50 of 41.8 nM).

CAS nr:

2133360-00-4

Purity:

98%

Molecular Weight:

771,78

SMILES:

O=C(NC1=CC=CC(C(N2C(CC3)C(NC3=O)=O)=O)=C1C2=O)COCCN4N=NC(CN5C(N(C)C6=C(C=C(C7=C(C)ON=C7C)C=C6)C5C8=CC=CC=C8)=O)=C4

Formula:

C40H37N9O8

Pathway:

Chromatin/Epigenetic

Target:

Epigenetic Reader Domain