Bioactivity:

RTS-V5 is a dual inhibitor of HDAC/proteasome (IC50s: 6.9, 18, 15, 0.27, 0.53 _M for HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, respectively).

CAS nr:

2285346-31-6

Purity:

98%

Molecular Weight:

525,6

SMILES:

O=C(NO)C1=CC=C(C(N[C@@H](CC(NCC(C)(C)C)=O)C(N[C@@H](C)C(NCC2=CC=CC=C2)=O)=O)=O)C=C1

Formula:

C27H35N5O6

Pathway:

DNA Damage/DNA Repair,Chromatin/Epigenetic

Target:

HDAC,HDAC