Bioactivity:

BIBO3304 TFA is an effective, orally active, and selective neuropeptide Y (NPY) Y1 receptor antagonist (IC50:0.38 and 0.72 nM for the human and the rat Y1 receptor).

CAS nr:

191868-14-1

Purity:

98%

Molecular Weight:

643,66

SMILES:

O=C(N[C@@H](C(NCC1=CC=C(CNC(N)=O)C=C1)=O)CCCNC(N)=N)C(C2=CC=CC=C2)C3=CC=CC=C3.O=C(O)C(F)(F)F

Formula:

C31H36F3N7O5

Pathway:

GPCR/G Protein,Neuroscience

Target:

Neuropeptide Y Receptor,Neuropeptide Y Receptor