Bioactivity:

BPK-29 is a specific ligand that disrupts the atypical orphan nuclear receptor NR0B1-protein interactions by covalently modifying C274. It impairs the anchorage-independent growth of KEAP1-mutant cancer cells.

CAS nr:

2143467-62-1

Purity:

98%

Molecular Weight:

470

SMILES:

O=C(N(C1CCN(C(C2=CC=C(N3CCOCC3)C=C2)=O)CCC1)CC4=CC=CC=C4)CCl

Formula:

C26H32ClN3O3

Pathway:

Others

Target:

Others