Bioactivity:

PF-06424439 methanesulfonate is an oral, potent and selective imidazopyridine diacylglycerol acyltransferase 2 (DGAT2) inhibitor(IC50 of 14 nM)[1]. PF-06424439 methanesulfonate is slowly reversible, time-dependent inhibitor, which inhibits DGAT2 in a nonc

CAS nr:

1469284-79-4

Purity:

98%

Molecular Weight:

536,05

SMILES:

O=C([C@H]1CN(C2=CC=C3C(NC(C4(N5N=CC(Cl)=C5)CC4)=N3)=N2)CCC1)N6CCCC6.CS(=O)(O)=O

Formula:

C23H30ClN7O4S

Pathway:

Metabolism,Metabolism,Proteases/Proteasome

Target:

Transferase,Acyltransferase,Acyltransferase