Bioactivity:

Men 10376 is a selective antagonist of tachykinin NK-2 receptor. It has a Ki of 4.4 _M for rat small intestine NK-2 receptor.

CAS nr:

135306-85-3

Purity:

98%

Molecular Weight:

1081,22

SMILES:

NCCCC[C@@H](C(N)=O)NC([C@@H](CC1=CNC2=C1C=CC=C2)NC([C@H](NC([C@H](C(C)C)NC([C@H](NC([C@@H](NC([C@@H](N)CC(O)=O)=O)CC3=CC=C(O)C=C3)=O)CC4=CNC5=C4C=CC=C5)=O)=O)CC6=CNC7=C6C=CC=C7)=O)=O

Formula:

C57H68N12O10

Pathway:

Cell Cycle/Checkpoint

Target:

CDK