Bioactivity:

PLX51107 is a potent and selective BET inhibitor (Kds: 1.6, 2.1, 1.7, and 5 nM for BRD2-BD1, BRD3-BD1, BRD4-BD1, and BRDT-BD1).

CAS nr:

1627929-55-8

Purity:

98%

Molecular Weight:

438,48

SMILES:

C[C@H](N1C=C(C2=C1C=C(C=N2)C1=C(C)ON=C1C)C1=CC=C(C=C1)C(O)=O)C1=CC=CC=N1

Formula:

C26H22N4O3

Pathway:

Chromatin/Epigenetic

Target:

Epigenetic Reader Domain