Bioactivity:

DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for _-, _-, and _-opioid receptors, respectively) with potent antinociceptive activity. DPI-3290 is one of a series of novel centrally acting agents.

CAS nr:

182417-73-8

Purity:

98%

Molecular Weight:

487,61

SMILES:

O=C(N(C1=CC=CC(F)=C1)C)C2=CC=CC([C@@H](N3[C@@H](C)CN(CC=C)[C@H](C)C3)C4=CC=CC(O)=C4)=C2

Formula:

C30H34FN3O2

Pathway:

Neuroscience,GPCR/G Protein,Endocrinology/Hormones

Target:

Opioid Receptor,Opioid Receptor,Opioid Receptor