Bioactivity:

SB-674042 is an effective and selective non-peptide orexin OX1 receptor antagonist (Kd = 3.76 nM). It exhibits 100-fold selectivity for OX1 over OX2 receptors.

CAS nr:

483313-22-0

Purity:

98%

Molecular Weight:

448,51

SMILES:

FC1=C(C2=C(C(N3[C@H](CC4=NN=C(C5=CC=CC=C5)O4)CCC3)=O)N=C(C)S2)C=CC=C1

Formula:

C24H21FN4O2S

Pathway:

Others

Target:

Others