MM 54 TP2001
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
Potent apelin receptor antagonist (Ki = 82 nM; IC50 = 93 nM). Antagonizes the inhibitory affect of [Pyr1]-Apelin-13 on forskolin-induced cAMP accumulation in CHO-K1-APJ cells. Recuces tumor expansion and lengthens survival time in a mouse xenograft model
CAS nr:
1313027-43-8
Purity:
98%
Molecular Weight:
1737,15
SMILES:
Formula:
C70H121N29O15S4
Pathway:
Target:
