Bioactivity:

Potent and selective melanocortin MC4 receptor antagonist (IC50 values are 11.63, 1115 and > 10 000 nM at MC4, MC3 and MC1 receptors respectively). Significantly reverses stress-induced anorexia but has no effect on food intake in free-feeding rats. Exhib

CAS nr:

475498-26-1

Purity:

98%

Molecular Weight:

609,73

SMILES:

CC(=O)N[C@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@H](Cc1ccc2ccccc2c1)C(N)=O

Formula:

C34H39N7O4

Pathway:

Neuroscience,GPCR/G Protein

Target:

Melanocortin Receptor,Melanocortin Receptor