Bioactivity:

TRV-120027 acetate is a _-arrestin-1-biased agonist of the angiotensin II receptor type 1 (AT1 receptor) and engages ﾧ-arrestins while blocking G-protein signaling.

CAS nr:

TP2158L1

Purity:

98%

Molecular Weight:

986,14

SMILES:

CC(O)=O.C[C@H](C(O)=O)NC([C@H]1N(C([C@H](CC2=CNC=N2)NC([C@H]([C@@H](C)CC)NC([C@H](CC3=CC=C(O)C=C3)NC([C@H](C(C)C)NC([C@H](CCCNC(N)=N)NC(CNC)=O)=O)=O)=O)=O)=O)CCC1)=O

Formula:

C45H71N13O12

Pathway:

Endocrinology/Hormones

Target:

RAAS