Bioactivity:

SNT-207858 free base is a selective, blood brain barrier penetrating, potent and orally active antagonist of melanocortin-4 (MC-4) receptor(IC50 of 22 nM (binding) and 11 nM (function), on the MC-4 receptor).

CAS nr:

1104662-66-9

Purity:

98%

Molecular Weight:

616,62

SMILES:

O=C(N1CCCC1)N[C@H](CC2=CC=C(Cl)C=C2Cl)C(N3CCC(C4=NC=CC=C4OC[C@H](N5CCCC5)CC)CC3)=O

Formula:

C32H43Cl2N5O3

Pathway:

Others

Target:

Others