Lifirafenib T22272
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
Lifirafenib is a potent inhibitor of RAF family kinases and EGFR in biochemical assays with IC50 of 23, 29 and 495 nM for the recombinant BRAFV600E kinase domain, EGFR and EGFR T790M/L858R mutant respectively.
CAS nr:
1446090-79-4
Purity:
98%
Molecular Weight:
478,42
SMILES:
O=C1Nc2nccc(Oc(cc3)cc(C45)c3OC4C5c3nc(ccc(C(F)(F)F)c4)c4[nH]3)c2CC1
Formula:
C25H17F3N4O3
Pathway:
MAPK,Tyrosine Kinase/Adaptors,Angiogenesis,JAK/STAT signaling
Target:
Raf,EGFR,EGFR,EGFR
