Bioactivity:

Fiboflapon is an orally bioavailable 5-lipoxygenase-activating protein (FLAP) inhibitor with a potency of 2.9 nM in FLAP binding, an IC50 of 76 nM for inhibition of LTB4 in human blood.

CAS nr:

936350-00-4

Purity:

98%

Molecular Weight:

637,83

SMILES:

CC(C(O)=O)(C)CC1=C(SC(C)(C)C)C2=CC(OCC3=CC=C(C)C=N3)=CC=C2N1CC4=CC=C(C5=CN=C(OCC)C=C5)C=C4

Formula:

C38H43N3O4S

Pathway:

Immunology/Inflammation

Target:

LTR