Bioactivity:

LPA2 antagonist 2 is _480-fold more selective than LPA3 (IC50 of 13.85 _M).LPA2 antagonist 2 is a selective LPA2 antagonist with an IC50 of 28.3 nM and a Ki of 21.1 nM.

CAS nr:

36840-10-5

Purity:

98%

Molecular Weight:

380,35

SMILES:

O=C(O)/C=C/C(NC1=CC=C(C2=CC=C(NC(/C=C/C(O)=O)=O)C=C2)C=C1)=O

Formula:

C20H16N2O6

Pathway:

GPCR/G Protein

Target:

LPA Receptor