ProTx III TP1969
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
Potent Nav1.7 blocker (IC50 = 2.5 nM). Also inhibits Nav1.1, Nav1.2, Nav1.3 and Nav1.6 in the nanomolar range. Exhibits no effects on Cav channels or nAChR at 5 _M. Demonstrates analgesic activity in vivo; antagonizes effects of scorpion-venom toxin OD1 a
CAS nr:
TP1969
Purity:
98%
Molecular Weight:
3802,41
SMILES:
Formula:
C162H246N52O43S6
Pathway:
Target:
