Avagacestat T6249
Specifications
| 1mg/5mg/10mg/25mg/50mg/100mg |
Bioactivity:
Avagacestat (BMS-708163) is a potent, selective, orally bioavailable _-secretase inhibitor of A_40 and A_42 with IC50 of 0.3 nM and 0.27 nM, demonstrating a 193-fold selectivity against Notch. Phase 2.
CAS nr:
1146699-66-2
Purity:
98%
Molecular Weight:
520,88
SMILES:
NC(=O)[C@@H](CCC(F)(F)F)N(CC1=C(F)C=C(C=C1)C1=NOC=N1)S(=O)(=O)C1=CC=C(Cl)C=C1
Formula:
C20H17ClF4N4O4S
Pathway:
Proteases/Proteasome,Neuroscience,Stem Cells
Target:
Gamma-secretase,Gamma-secretase,Gamma-secretase
