Bioactivity:

ERK1/2 inhibitor 1 is a potent, orally bioavailable ERK1/2 inhibitor, showing 60% inhibition at 1 nM and an IC50 of 3.0 nM against ERK1 and ERK2, respectively.

CAS nr:

2095719-90-5

Purity:

98%

Molecular Weight:

550,05

SMILES:

ClC1=CN=C(NC2CCOCC2)N=C1C3=CC=C(CN([C@H](C)C(N[C@H](CO)C4=CC=CC(C)=C4)=O)C5=O)C5=C3

Formula:

C29H32ClN5O4

Pathway:

MAPK

Target:

ERK