JNJ-5207852 dihydrochloride M22976
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Specifications
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CAS Number:
1782228-76-5
Target:
Histamine Receptor
Molecular formula:
C20H34Cl2N2O
Formula weight:
389,4
Purity:
>98% (HPLC)
Stability:
≥ 2 years
Product description:
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor. JNJ-5207852 is a potent dibasic amine antagonist that binds potently to rat H3 receptors (Ki=1.2 nm), and has good brain penetration. In ex vivo binding studies in mice, the compound had an ED50 of 0.13 mg kg−1, subcutaneously.
Note:
Research use only, not for human use.
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