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GSK2807 Trifluoroacetate M22934



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Specifications

inquiry

CAS Number:

2245255-66-5

Target:

Other Targets

Molecular formula:

C21H33F3N8O7

Formula weight:

566,53

Purity:

>98% (HPLC)

Stability:

≥ 2 years

Product description:

GSK2807 Trifluoroacetate is a selective and SAM-competitive inhibitor of SMYD3 (Ki: 14 nM; IC50: 130 nM).GSK2807, a potent and selective, SAM-competitive inhibitor of SMYD3 (Ki = 14 nM). A high-resolution crystal structure reveals that GSK2807 bridges the gap between the SAM-binding pocket and the substrate lysine tunnel of SMYD3.

Note:

Research use only, not for human use.

More info:

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