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UT-34 M22452



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Specifications

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CAS Number:

2168525-92-4

Target:

Androgen Receptor

Molecular formula:

C15H12F4N4O2

Formula weight:

356,27

Purity:

>98% (HPLC)

Stability:

≥ 2 years

Product description:

UT-34 is a selective and orally active antagonist of second-generation pan-androgen receptor (AR) and degrader(IC50s of 211.7 nM, 262.4 nM and 215.7 nM for wild-type, F876L and W741L AR, respectively), and has anti-prostate cancer efficacy. In LNCaP cells, UT-34 (3-10 µM; 24 hours) treatment inhibits the expression of PSA and FKBP5 and growth of LNCaP cells starting from 100 nM with maximum effect observed at 10 μM.

Note:

Research use only, not for human use.

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