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AMG-548 M16264



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Specifications

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CAS Number:

864249-60-5

Target:

p38 MAPK

Molecular formula:

C29H27N5O

Formula weight:

461,569

Purity:

>98% (HPLC)

Stability:

≥ 2 years

Product description:

AMG-548 is a potent and selective inhibitor of p38α with Ki of 0.5 nM, dispalys weak inhibition for p38β (Ki=3.6 nM), and >5,000-fold selectivity over p38γ and p38δ; shows >1,000-fold selectivity over other 36 kinases, and is efficacious in acute and chronic models of arthritis. Rheumatoid ArthritisDiscontinued

Note:

Research use only, not for human use.

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